CNS Pharmacology Review 10 June :22 AM
Acetaminophen Analgesic, Antipyretic
Adrenocorticotropin (ACTH) Anterior pituitary hormone Anticonvulsant Stimulates synthesis and release of cortisol
Alfentanil Opioid General anaesthetic Intravenous anaesthetic
Amantadine Antiviral Antiparkinson Treatment of Influenza A Inhibits replication at the stage of uncoating Inhibits dopamine release
Amitriptyline Tricyclic antidepressant (TCA)
Amphetamine Indirect sympathomimetic Drug of abuse ADD treatment Stimulant
Atropine Anticholinergic Antimuscarinic Treatment for bradycardia, diarrhea, cholinesterase poisoning
Baclofen Skeletal muscle relaxant Anxiolytic GABA B agonist
Benztropine Anticholinergic Antiparkinson Muscarinic receptor antagonist
Bethanecol Cholinomimetic Muscarinic agonist Induces defecation and urination Bronchoconstrictor
Bromocriptine Antiparkinson Dopamine (D 2 ) agonist Inhibits prolactin release
Brupropion Second generation antidepressant
Buprenorphine Opioid Partial agonist
Buspirone Sedative/hypnotic Anxiolytic
Butorphanol Opioid Analgesic receptor partial agonist or antagonist
Carbamazepine Anticonvulsant
Carbidopa Antiparkinson Peripheral dopa decarboxylase inhibitor
Celecoxib NSAID Anti-inflammatory Cyclooxygenase 2 (COX-2) inhibitor
Chloral hydrate Sedative/Hypnotic General anaesthetic Acts on GABA A receptor complex Similar to barbiturates
Chlordiazepoxide Sedative/hypnotic Anxiolytic Benodiazepine Acts on GABA A receptor complex
Chlorpromazine Antipsychotic Phenothiazine
Clozapine Antipsychotic
Cocaine Indirect sympathomimetic Drug of abuse Topical anaesthetic Stimulant Local anaesthetic
Codeine Opioid Analgesic Weak agonist
Dantrolene Skeletal muscle relaxant Ryanodine receptor antagonist Treatment for malignant hyperthermia
Deprenyl/selegiline Antiparkinson Monoamine oxidase B inhibitor (MAO-I) Potentiates effects of L-Dopa
Desipramine Tricyclic antidepressant (TCA)
Dextromethorphan Opioid Antitussive
Diazepam Sedative/hypnotic Anxiolytic Anticonvulsant Benzodiazepine Acts on GABA A receptor complex
Diflunisal NSAID Analgesic, Anti-inflammatory Antipyretic Cyclooxygenase inhibitor
Diphenoxylate docusate Antidiarrheal Opiate
Enflurane General anaesthetic Inhaled anaesthetic
Entacapone Antiparkinson Peripheral catechol-o- methyltransferase inhibitor
Ephedra (Ma Huang) Dietary supplement Amphetamine-like stimulant
Ethanol Drug of abuse Sedative
Ethosuximide Anticonvulsant
Etomidate General anaesthetic Intravenous anaesthetic
Fentanyl Opioid Analgesic receptor agonist
Flumazenil Benzodiazepine antagonist Acts on GABA A receptor complex
Fluoxetine Antidepressant Selective serotonin reuptake inhibitor (SSRI)
Flurazepam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
Ginko biloba Dietary supplement Treatment of Alzheimer symptoms
Glutethimide Sedative/Hypnotic
Haloperidol Antipsychotic
Halothane General anaesthetic Inhaled anaesthetic
Heroin Drug of abuse Opioid
Imipramine Indirect sympathomimetic Tricyclic antidepressant (TCA) Antimicturant
Indomethacin NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor Tocolytic Uterine relaxant
Isoflurane General anaesthetic Inhaled anaesthetic
Kava kava Dietary supplement Stress relief and treatment of insomnia
Ketamine General anaesthetic Drug of abuse Sedative
Ketoprofen NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
Levodopa Antiparkinson Dopamine precursor
Lidocaine Class I antiarrhythmic Local anaesthetic Na + channel blocker (activated and inactivated channels)
Lithium Antidepressant Used to treat manic/depressive disorder
Loperamide Antidiarrheal Opiate
Lorazepam Anxiolytic Anticonvulsant Benzodiazepine Acts on GABA A receptor complex
Lysergic acid diethylamide (LSD) Drug of abuse Hallucinogen
Marijuana Drug of abuse Cannabinoid
Meperidine Opioid analgesic receptor agonist
Mepivacaine Local anaesthetic
Meprobamate Sedative/hypnotic Anxiolytic
Meclofenamate NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
Metamphetamine Drug of abuse Stimulant
Methadone Opioid receptor agonist
Morphine Opioid Analgesic receptor agonist
Nalbuphine Opioid antagonist receptor antagonist
Nalmefene Opioid antagonist
Nalorphine Opioid antagonist
Naloxone Opioid antagonist
Naltrexone Opioid antagonist
Naproxen NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
Neostigmine Anticholinesterase Vasodilator Treatment for myaesthenia gravis Promotes defecation and urination Bronchoconstrictor
Nicotine Cholinomimetic Drug of abuse Nicotinic receptor agonist (skeletal muscle contraction) Stimulant Smoking cessation medication
Nitrous oxide General anaesthetic Inhaled anaesthetic
Non-steroidal Anti-inflammatory Drugs (NSAIDs) Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitors
Nortriptyline Tricyclic antidepressant (TCA)
Oxazepam Sedative/hypnotic Anxiolytic Benzodiazepine Acts on GABA A receptor complex
Oxybutinin Anticholinergic Muscarinic receptor antagonist Prevents urination
Oxycodone Analgesic Opioid agonist
Paraldehyde Sedative/Hypnotic
Pentazocine Opioid analgesic receptor partial agonist or antagonist
Pentobarbital Sedative/Hypnotic Barbiturate
Phencyclidine (PCP) Drug of abuse Hallucinogen
Phenobarbital Sedative/Hypnotic Anticonvulsant Barbiturate
Phenytoin Anticonvulsant Class I antiarrhythmic Na + channel blocker (inactivated channels)
Piroxicam NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
Pramipexole Antiparkinson Dopamine agonist (non-ergot)
Primidone Anticonvulsant
Procaine Local anaesthetic
Propofol General anaesthetic Intravenous anaesthetic
Resperidone Antipsychotic
Ropinirole Antiparkinson Dopamine agonist (non-ergot)
Sertraline Antidepressant Selective serotonin reuptake inhibitor (SSRI)
Sildenafil Vasodilator Promotes erection
St. John’s Wort Dietary supplement Antidepressant
Sufentanil Opioid General anaesthetic Intravenous anaesthetic
Sulindac NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
Temazepam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
Tetracaine Local anaesthetic
Thiopental General anaesthetic Ultra-short-acting barbiturate
Thioridazine Antipsychotic Phenothiazine
Thiothixene Antipsychotic
Tolterodine Anticholinergic Muscarinic receptor antagonist Prevents urination
Tranylcypromine Antidepressant Monoamine oxidase inhibitor (MAO-I)
Triazolam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
Trifluoperazine Antipsychotic Phenothiazine
Trihexyphenidyl Antiparkinson Antimuscarinic
Valproic acid Anticonvulsant
Vigabatrin Anticonvulsant Irreversible GABA aminotransferase inhibitor
Zolpidem Sedative/Hypnotic Non-benzodiazepine