Cardiovascular System Pharmacology Review 23 November :24 AM
Acebutolol Sympatholytic 1 adrenergic antagonist Antihypertensive Antianginal Antiarrhythmic Bronchoconstrictor
Acetylcholine Cholinomimetic Antigluacoma Muscle contraction (nicotinic receptor)
Adenosine Antiarrhythmic Miscellaneous (does not fit class I-IV organization)
Albuterol Sympathomimetic 2 adrenergic agonist Short acting bronchodilator Used in asthma
Amiodarone Class I/III antiarrhythmic Na + and K + channel blocker (inactivated channels)
Amphetamine Indirect sympathomimetic Drug of abuse ADD treatment Stimulant
Amyl nitrite Vasodilator Antianginal Aerosol
Angiotensin II Autacoid Vasoconstrictor
Atenolol Sympatholytic 1 adrenergic antagonist Antihypertensive Antiarrhythmic Antianginal Bronchoconstrictor
Atorvastatin Antihyperlipidemic HMG-CoA reductase inhibitor
Atropine Anticholinergic Antimuscarinic Treatment for bradycardia, diarrhea, cholinesterase poisoning
Betaxolol Sympatholytic 1 adrenergic antagonist Antihypertensive Glaucoma medication Bronchoconstrictor
Bethanecol Cholinomimetic Muscarinic agonist Induces defecation and urination Bronchoconstrictor
Biltolterol Sympathomimetic 2 adrenergic agonist Bronchodilator
Bretylium Sympatholytic Class III antiarrhythmic K + channel blocker
Candesartan Antihypertensive Angiotensin receptor blocker (ARB)
Captopril Antihypertensive Converting enzyme inhibitor Heart failure treatment Angioedema producer
Cholestyramine Antihyperlipidemic Bile acid binding resin (BABR)
Clofibrate Antihyperlipidemic Lipoprotein lipase activator
Clonidine Sympatholytic 2 adrenergic agonist Antihypertensive
Colestipol Antihyperlipidemic Bile acid binding resin (BABR)
Diazoxide Vasodilator Antihypertensive
Digitalis Cardiac glycoside Antiarrhythmic Na + /K + ATPase inhibitor Positive inotrope Miscellaneous (does not fit class I-IV organization)
Digitoxin Cardiac glycoside Antiarrhythmic Na + /K + ATPase inhibitor Positive inotrope Miscellaneous (does not fit class I-IV organization)
Digoxin Cardiac glycoside Antiarrhythmic Na + /K + ATPase inhibitor Positive inotrope Miscellaneous (does not fit class I-IV organization)
DIG-specific antibody fragments Antidote Cardiac glycoside poisoning
Diltiazem Class IV antiarrhythmic Antihypertensive Ca 2+ channel blocker
Disopyramide Class I antiarrhythmic Na + channel blocker (activated channels)
Dobutamine Sympathomimetic 1 adrenergic agonist Inotrope
Dofetilide Class III antiarrhythmic K + channel blocker
Dopamine Sympathomimetic Inotrope Vasodilator
Doxazosin Sympatholytic 1 adrenergic antagonist Antihypertensive
Ecothiophate Anticholinesterase Vasodilator Bronchoconstrictor Glaucoma treatment
Edrophonium Anticholinesterase Vasodilator Diagnostic for myaesthenia gravis Bronchoconstrictor
Enalapril Antihypertensive Converting enzyme inhibitor Angioedema producer
Ephedrine Indirect sympathomimetic Vasoconstrictor Bronchodilator Decongestant
Epinephrine Sympathomimetic and adrenergic agonist Vasoconstrictor Bronchodilator
Eprosartan Antihypertensive Angiotensin receptor blocker (ARB)
Esmolol Sympatholytic 1 adrenergic antagonist Class II Antiarrhythmic Antihypertensive Bronchoconstrictor
Ezitimibe Antihyperlipidemic Cholesterol absorption inhibitor
Fenofibrate Antihyperlipidemic Lipoprotein lipase activator
Flecainide Class I antiarrhythmic Na + channel blocker
Fluvastatin Antihyperlipidemic HMG-CoA Reductase Inhibitor
Fosinopril Antihypertensive Converting enzyme inhibitor
Gemfibrozil Antihyperlipidemic Lipoprotein lipase activator
Guanabenz Sympatholytic Antihypertensive
Guanadrel Sympatholytic Antihypertensive
Guanethidine Sympatholytic Antihypertensive
Guanfacine Sympatholytic 2 adrenergic agonist Antihypertensive
Hydralazine Vasodilator Antihypertensive
Ibutilide Class III antiarrhythmic K + channel blocker
Imipramine Indirect sympathomimetic Tricyclic antidepressant (TCA) Antimicturant
Isoproterenol Sympathomimetic adrenergic agonist Vasodilator Bronchodilator
Isosorbide dinitrate Venodilator Used to treat CHF
Lidocaine Class I antiarrhythmic Local anaesthetic Na + channel blocker (activated and inactivated channels)
Lisinopril Antihypertensive Converting enzyme inhibitor Heart failure treatment Angioedema producer
Losartan Antihypertensive Angiotensin receptor blocker (ARB)
Lovastatin Antihyperlipidemic HMG-CoA reductase inhibitor
Malathion Anticholinesterase Vasodilator Bronchoconstrictor
Metaproterenol Sympathomimetic 2 adrenergic agonist Bronchodilator Used in asthma
Methacholine Cholinomimetic Bronchoconstrictor
Methoxamine Sympathomimetic 1 adrenergic agonist Vasoconstrictor
Methydopa Sympatholytic 2 adrenergic agonist Antihypertensive
Methylphenidate Indirect sympathomimetic Drug of abuse ADD treatment Stimulant
Metoprolol Sympatholytic 1 adrenergic antagonist Antihypertensive Heart failure medication Bronchoconstrictor
Mexilitine Class I antiarrhythmic Na + channel blocker (activated and inactivated channels)
Minoxidil Vasodilator Antihypertensive
Moezipril Antihypertensive Converting enzyme inhibitor
Moricizine Class I antiarrhythmic Na + channel blocker
Nadolol Sympatholytic adrenergic antagonist Antihypertensive
Neostigmine Anticholinesterase Vasodilator Treatment for myaesthenia gravis Promotes defecation and urination Bronchoconstrictor
Nicotine Cholinomimetic Drug of abuse Nicotinic receptor agonist (skeletal muscle contraction) Stimulant Smoking cessation medication
Nicotinic acid Antihyperlipidemic Inhibition of VLDL secretion (?)
Nifedipine Antihypertensive Antianginal Calcium channel blocker
Nitroglycerine Venodilator Antianginal
Nitroprusside Vasodilator Antihypertensive
Norepinephrine Sympathomimetic Vasoconstrictor
Perindopril Antihypertensive Converting enzyme inhibitor
Phenoxybenzamine Sympatholytic adrenergic antagonist Antihypertensive
Phentolamine Sympatholytic adrenergic antagonist Antihypertensive
Phenylephrine Sympathomimetic 1 adrenergic agonist Vasoconstrictor Nasal decongestant
Phenytoin Anticonvulsant Class I antiarrhythmic Na + channel blocker (inactivated channels)
Physostigmine Anticholinesterase Bradycardic Vasodilator Bronchoconstrictor
Pilocarpine Cholinomimetic Muscarinic agonist Antiglaucoma Bronchoconstrictor
Pindolol Sympatholytic adrenergic antagonist Antihypertensive Bronchoconstrictor
Pravastatin Antihyperlipidemic HMG-CoA reductase inhibitor
Prazosin Sympatholytic 1 adrenergic antagonist Antihypertensive
Propranolol Sympatholytic adrenergic antagonist Class II antiarrhythmic Antihypertensive Bronchoconstrictor
Pseudoephedrine Sympathomimetic and adrenergic agonist Vasoconstrictor Nasal decongestant
Pyridostigmine Anticholinesterase Vasodilator Treatment for myaesthenia gravis Bronchoconstrictor
Quinapril Antihypertensive Converting enzyme inhibitor
Quinidine Antimalarial Protein and nucleic acid synthesis inhibitor Class I antiarrhythmic Intercalates in DNA Binds to ferriprotoporphyrin Na + channel blocker
Ramipril Antihypertensive Converting enzyme inhibitor
Reserpine Sympatholytic Antihypertensive
Sildenafil Vasodilator Promotes erection
Simvastatin Antihyperlipidemic HMG-CoA reductase inhibitor
Sotolol Class II antiarrythmic Sympatholytic adrenergic antagonist
Terazosin Sympatholytic 1 adrenergic antagonist Antihypertensive Treatment for benign prostatic hypertrophy
Terbutaline Sympathomimetic 2 adrenergic agonist Short acting bronchodilator Tocolytic Uterine relaxant
Timolol Sympatholytic adrenergic antagonist Antihypertensive Glaucoma treatment Anti-anginal Bronchoconstrictor
Tocainide Class I antiarrhythmic Na + channel blocker (activated channels)
Trandopril Antihypertensive Converting enzyme inhibitor
Trimethaphan Sympatholytic Anticholinergic Nicotinic antagonist Antihypertensive
Tyramine Indirect sympathomimetic Vasoconstrictor Vasopressor
Valsartan Antihypertensive Angiotensin receptor blocker (ARB)
Verapamil Class IV antiarrhythmic Antihypertensive L-type Ca 2+ channel blocker Antianginal