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Enzyme flexibility, solvent and weak interactions characterize thrombin–ligand interactions: implications for drug design Richard A Engh, Hans Brandstetter,

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Presentation on theme: "Enzyme flexibility, solvent and weak interactions characterize thrombin–ligand interactions: implications for drug design Richard A Engh, Hans Brandstetter,"— Presentation transcript:

1 Enzyme flexibility, solvent and weak interactions characterize thrombin–ligand interactions: implications for drug design Richard A Engh, Hans Brandstetter, Gudrun Sucher, Andreas Eichinger, Ulrich Baumann, Wolfram Bode, Robert Huber, Thomas Poll, Rainer Rudolph, Wolfgang von der Saal Structure Volume 4, Issue 11, Pages 1353-1362 (November 1996) DOI: 10.1016/S0969-2126(96)00142-6

2 Figure 1 Structure 1996 4, 1353-1362DOI: (10.1016/S0969-2126(96)00142-6)

3 Figure 2 Structure 1996 4, 1353-1362DOI: (10.1016/S0969-2126(96)00142-6)

4 Figure 3 Structure 1996 4, 1353-1362DOI: (10.1016/S0969-2126(96)00142-6)

5 Figure 4 Structure 1996 4, 1353-1362DOI: (10.1016/S0969-2126(96)00142-6)

6 Figure 5 Structure 1996 4, 1353-1362DOI: (10.1016/S0969-2126(96)00142-6)

7 Figure 6 Structure 1996 4, 1353-1362DOI: (10.1016/S0969-2126(96)00142-6)

8 Figure 7 Structure 1996 4, 1353-1362DOI: (10.1016/S0969-2126(96)00142-6)


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