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2003-2004 CNS Pharmacology Review 10 June 2015 2:22 AM
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Acetaminophen Analgesic, Antipyretic
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Adrenocorticotropin (ACTH) Anterior pituitary hormone Anticonvulsant Stimulates synthesis and release of cortisol
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Alfentanil Opioid General anaesthetic Intravenous anaesthetic
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Amantadine Antiviral Antiparkinson Treatment of Influenza A Inhibits replication at the stage of uncoating Inhibits dopamine release
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Amitriptyline Tricyclic antidepressant (TCA)
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Amphetamine Indirect sympathomimetic Drug of abuse ADD treatment Stimulant
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Atropine Anticholinergic Antimuscarinic Treatment for bradycardia, diarrhea, cholinesterase poisoning
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Baclofen Skeletal muscle relaxant Anxiolytic GABA B agonist
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Benztropine Anticholinergic Antiparkinson Muscarinic receptor antagonist
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Bethanecol Cholinomimetic Muscarinic agonist Induces defecation and urination Bronchoconstrictor
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Bromocriptine Antiparkinson Dopamine (D 2 ) agonist Inhibits prolactin release
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Brupropion Second generation antidepressant
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Buprenorphine Opioid Partial agonist
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Buspirone Sedative/hypnotic Anxiolytic
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Butorphanol Opioid Analgesic receptor partial agonist or antagonist
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Carbamazepine Anticonvulsant
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Carbidopa Antiparkinson Peripheral dopa decarboxylase inhibitor
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Celecoxib NSAID Anti-inflammatory Cyclooxygenase 2 (COX-2) inhibitor
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Chloral hydrate Sedative/Hypnotic General anaesthetic Acts on GABA A receptor complex Similar to barbiturates
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Chlordiazepoxide Sedative/hypnotic Anxiolytic Benodiazepine Acts on GABA A receptor complex
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Chlorpromazine Antipsychotic Phenothiazine
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Clozapine Antipsychotic
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Cocaine Indirect sympathomimetic Drug of abuse Topical anaesthetic Stimulant Local anaesthetic
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Codeine Opioid Analgesic Weak agonist
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Dantrolene Skeletal muscle relaxant Ryanodine receptor antagonist Treatment for malignant hyperthermia
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Deprenyl/selegiline Antiparkinson Monoamine oxidase B inhibitor (MAO-I) Potentiates effects of L-Dopa
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Desipramine Tricyclic antidepressant (TCA)
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Dextromethorphan Opioid Antitussive
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Diazepam Sedative/hypnotic Anxiolytic Anticonvulsant Benzodiazepine Acts on GABA A receptor complex
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Diflunisal NSAID Analgesic, Anti-inflammatory Antipyretic Cyclooxygenase inhibitor
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Diphenoxylate docusate Antidiarrheal Opiate
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Enflurane General anaesthetic Inhaled anaesthetic
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Entacapone Antiparkinson Peripheral catechol-o- methyltransferase inhibitor
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Ephedra (Ma Huang) Dietary supplement Amphetamine-like stimulant
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Ethanol Drug of abuse Sedative
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Ethosuximide Anticonvulsant
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Etomidate General anaesthetic Intravenous anaesthetic
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Fentanyl Opioid Analgesic receptor agonist
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Flumazenil Benzodiazepine antagonist Acts on GABA A receptor complex
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Fluoxetine Antidepressant Selective serotonin reuptake inhibitor (SSRI)
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Flurazepam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
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Ginko biloba Dietary supplement Treatment of Alzheimer symptoms
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Glutethimide Sedative/Hypnotic
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Haloperidol Antipsychotic
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Halothane General anaesthetic Inhaled anaesthetic
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Heroin Drug of abuse Opioid
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Imipramine Indirect sympathomimetic Tricyclic antidepressant (TCA) Antimicturant
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Indomethacin NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor Tocolytic Uterine relaxant
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Isoflurane General anaesthetic Inhaled anaesthetic
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Kava kava Dietary supplement Stress relief and treatment of insomnia
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Ketamine General anaesthetic Drug of abuse Sedative
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Ketoprofen NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Levodopa Antiparkinson Dopamine precursor
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Lidocaine Class I antiarrhythmic Local anaesthetic Na + channel blocker (activated and inactivated channels)
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Lithium Antidepressant Used to treat manic/depressive disorder
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Loperamide Antidiarrheal Opiate
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Lorazepam Anxiolytic Anticonvulsant Benzodiazepine Acts on GABA A receptor complex
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Lysergic acid diethylamide (LSD) Drug of abuse Hallucinogen
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Marijuana Drug of abuse Cannabinoid
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Meperidine Opioid analgesic receptor agonist
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Mepivacaine Local anaesthetic
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Meprobamate Sedative/hypnotic Anxiolytic
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Meclofenamate NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Metamphetamine Drug of abuse Stimulant
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Methadone Opioid receptor agonist
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Morphine Opioid Analgesic receptor agonist
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Nalbuphine Opioid antagonist receptor antagonist
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Nalmefene Opioid antagonist
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Nalorphine Opioid antagonist
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Naloxone Opioid antagonist
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Naltrexone Opioid antagonist
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Naproxen NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Neostigmine Anticholinesterase Vasodilator Treatment for myaesthenia gravis Promotes defecation and urination Bronchoconstrictor
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Nicotine Cholinomimetic Drug of abuse Nicotinic receptor agonist (skeletal muscle contraction) Stimulant Smoking cessation medication
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Nitrous oxide General anaesthetic Inhaled anaesthetic
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Non-steroidal Anti-inflammatory Drugs (NSAIDs) Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitors
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Nortriptyline Tricyclic antidepressant (TCA)
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Oxazepam Sedative/hypnotic Anxiolytic Benzodiazepine Acts on GABA A receptor complex
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Oxybutinin Anticholinergic Muscarinic receptor antagonist Prevents urination
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Oxycodone Analgesic Opioid agonist
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Paraldehyde Sedative/Hypnotic
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Pentazocine Opioid analgesic receptor partial agonist or antagonist
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Pentobarbital Sedative/Hypnotic Barbiturate
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Phencyclidine (PCP) Drug of abuse Hallucinogen
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Phenobarbital Sedative/Hypnotic Anticonvulsant Barbiturate
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Phenytoin Anticonvulsant Class I antiarrhythmic Na + channel blocker (inactivated channels)
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Piroxicam NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Pramipexole Antiparkinson Dopamine agonist (non-ergot)
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Primidone Anticonvulsant
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Procaine Local anaesthetic
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Propofol General anaesthetic Intravenous anaesthetic
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Resperidone Antipsychotic
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Ropinirole Antiparkinson Dopamine agonist (non-ergot)
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Sertraline Antidepressant Selective serotonin reuptake inhibitor (SSRI)
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Sildenafil Vasodilator Promotes erection
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St. John’s Wort Dietary supplement Antidepressant
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Sufentanil Opioid General anaesthetic Intravenous anaesthetic
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Sulindac NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Temazepam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
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Tetracaine Local anaesthetic
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Thiopental General anaesthetic Ultra-short-acting barbiturate
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Thioridazine Antipsychotic Phenothiazine
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Thiothixene Antipsychotic
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Tolterodine Anticholinergic Muscarinic receptor antagonist Prevents urination
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Tranylcypromine Antidepressant Monoamine oxidase inhibitor (MAO-I)
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Triazolam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
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Trifluoperazine Antipsychotic Phenothiazine
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Trihexyphenidyl Antiparkinson Antimuscarinic
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Valproic acid Anticonvulsant
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Vigabatrin Anticonvulsant Irreversible GABA aminotransferase inhibitor
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Zolpidem Sedative/Hypnotic Non-benzodiazepine
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