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2004-2005 Pharmacology Review of Everything (Principles, Cardiovascular and Respiratory drugs have been updated) 26 October 2015 4:15 AM
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Hydrochlorothiazide Thiazide diuretic Na-Cl symporter inhibitor Antihypertensive
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Hydrocortisone Adrenocorticosteroid Glucocorticoid Anti-inflammatory steroid
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Hydroxychloroquine Disease modifying anti-rheumatic drug (DMARD)
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4-Hydroxycoumarin Oral anticoagulant Vitamin K synthesis inhibitor
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Hydroxyurea Antineoplastic Miscellaneous Ribonucleotide reductase inhibitor
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Hydroxyzine Classical antihistamine H 1 antagonist
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Ibritumomab Antineoplastic Anti-CD20 antibody
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Ibuprofen NSAID Analgesic, Anti-inflammatory Antipyretic Reversible cyclooxygenase inhibitor
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Ibutilide Class III antiarrhythmic K + channel blocker
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Imatinib Antineoplastic Miscellaneous Tyrosine kinase inhibitor
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Imipenem/Cilastatin New lactam antibiotic Cilastatin inhibits a kidney dipeptidase that inactivates imipenem
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Imipramine Indirect sympathomimetic Tricyclic antidepressant (TCA) Antimicturant
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Indapamide Thiazide-like diuretic Na-Cl symporter inhibitor Antihypertensive
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Indinavir Antiretroviral Protease inhibitor (PI)
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Indomethacin NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor Tocolytic Uterine relaxant
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Infliximab TNF inhibitor Anti-TNF monoclonal antibody Treatment of IBD
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Insulin Hormone Insulin analogue Short acting
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Interferon alpha Antiviral for hepatitis Antineoplastic Cytokine Anti-angiogenesis
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Interleukin 2 Cytokine Antineoplastic
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Interleukin 11 Cytokine Antineoplastic (supporting agent)
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Iodide Antithyroid Prevents synthesis and release of thyroid hormones (blocks iodine organification) Decreases hyperplasia
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Iodoquinol Antiparasitic Treatment of protozoal infections
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Ipecac Emetic
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Ipratropium Anticholinergic Antimuscarinic Inhaled bronchodilator
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Irbesartan Antihypertensive Angiotensin receptor blocker (ARB)
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Iressa Antineoplastic Miscellaneous Tyrosine kinase inhibitor
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Irinotecan Antineoplastic Natural product
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Iron (ferrous sulfate, iron dextran) Essential nutrient Required for hemoglobin and myoglobin synthesis
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Isoetharine Sympathomimetic adrenergic agonist Bronchodilator
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Isoflurane General anaesthetic Inhaled anaesthetic
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Isoniazid Antibiotic Inhibits biosynthesis of mycolic acids Major drug for tuberculosis
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Isoproterenol Sympathomimetic adrenergic agonist Vasodilator Bronchodilator
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Isosorbide dinitrate Venodilator Used to treat CHF
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Isradipine Antihypertensive Calcium channel blocker
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Itraconazole Triazole antifungal Inhibits synthesis of ergosterol by inhibiting lanosterol 14 demethylase
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Ivermectin Antihelminthic Treatment of intestinal and tissue roundworms
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Kallidin Inflammatory mediator Plasma, hypotension, pain
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Kaolin Antidiarrheal
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Kava kava Dietary supplement Stress relief and treatment of insomnia
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Ketamine General anaesthetic Drug of abuse Sedative
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Ketoconazole Imidazole antifungal Inhibits synthesis of ergosterol by inhibiting lanosterol 14 demethylase
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Ketoprofen NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Labetalol Sympatholytic and adrenergic antagonist Antihypertensive
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Lactulose Saline (osmotic) cathartic
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Lamivudine Antiretroviral Nucleoside reverse transcriptase inhibitor (NRTI)
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Lansoprazole Antiulcer H + /K + ATPase inhibitor
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Lente insulin Hormone Insulin analogue Intermediate acting
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Lepirudin Anticoagulant Direct thrombin inhibitor (DTI)
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Letrozole Antineoplastic Antiestrogen Aromatase Inhibitor
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Leukotriene B 4 (LTB 4 ) Inflammatory mediator Lipoxygenase product of arachidonate metabolism Chemotactic
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Leukotrienes C 4, D 4, E 4 (LTC 4, LTD 4, LTE 4 ) Inflammatory mediators Cysteinyl leukotrienes Peptidyl leukotrienes SRS-A Lipoxygenase products of arachidonate metabolism
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Leucovorin Antineoplastic (supporting agent) Folic acid analogue (used in methotrexate rescue)
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Leuprolide Antineoplastic Gonadotropin releasing hormone (GnRH) agonist
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Levobunolol Sympatholytic adrenergic antagonist Antihypertensive Bronchoconstrictor
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Levodopa Antiparkinson Dopamine precursor Inhibits growth hormone release
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Levonorgestrel Progestin 19-nor testosterone analogue Combination oral contraceptive
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Levothyroxine (T 4 ) Thyroid hormone
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Lidocaine Class I antiarrhythmic Local anaesthetic Na + channel blocker (activated and inactivated channels)
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Linezolid Oxazolidinone antibiotic Protein synthesis inhibitor 50S ribosomal subunit
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Liothyronine (T 3 ) Thyroid hormone
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Lisinopril Antihypertensive Converting enzyme inhibitor Heart failure treatment Angioedema producer
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Lispro insulin Hormone Insulin analogue Ultra short acting
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Lithium Antidepressant Used to treat manic/depressive disorder
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Lomustine (CCNU) Antineoplastic Alkylating agent Nitrosourea
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Loperamide Antidiarrheal Opiate
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Loratidine Antihistamine H 1 antagonist Non-sedating
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Lorazepam Anxiolytic Anticonvulsant Benzodiazepine Acts on GABA A receptor complex
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Losartan Antihypertensive Angiotensin receptor blocker (ARB)
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Lovastatin Antihyperlipidemic HMG-CoA reductase inhibitor
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Lutenizing Hormone (LH) Anterior pituitary hormone Regulator of gonadal function
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Lypressin Antidiuretic hormone analogue
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Lysergic acid diethylamide (LSD) Drug of abuse Hallucinogen
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Macrolides erythromycin, azithromycin, clarithromycin Antibiotics Bacteriostatic protein synthesis inhibitors 50S ribosome
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Magnesium hydroxide Antiulcer Saline (osmotic) cathartic Antacid
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Magnesium sulfate Calcium antagonist Tocolytic Uterine relaxant
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Malathion Anticholinesterase Vasodilator Bronchoconstrictor
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Mannitol Osmotic diuretic
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Marijuana Drug of abuse Cannabinoid
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Mebendazole Antihelminthic Treatment of intestinal roundworms
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Meclizine Antihistamine Antiemetic H 1 receptor antagonist
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Meclofenamate NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Mechlorethamine Antineoplastic Alkylating agent Nitrogen mustard
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Medroxyprogesterone Progestin Synthetic progesterone analogue Contraceptive
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Mefloquine Antimalarial Treatment and prophylaxis for chloroquine resistant Plasmodium
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Meglumine antimonate Tropical antiparasitic Organic antimonial Treatment of Leishmaniasis
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Melarsoprol Tropical antiparasitic Treatment of African Trypanosomiasis in CNS
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Melphalan Antineoplastic Alkylating agent Nitrogen mustard
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Menotropin Hormone Gonadotropin Ovulation inducing agent
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Meperidine Opioid analgesic receptor agonist
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Mepivacaine Local anaesthetic
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Meprobamate Sedative/hypnotic Anxiolytic
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6-Mercaptopurine Antineoplastic Antimetabolite (“pseudofeedback inhibition” of HGPRT and PRP – purine synthesis)
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Mesalamine (5-ASA) NSAID (salicylate) Treatment of IBD
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Mesna Antineoplastic (supporting agent) Prevent hemorrhagic cystitis due to cyclophosphamide
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Mestranol Estrogen Synthetic female gonadal steroid Combination oral contraceptive
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Metamphetamine Drug of abuse Stimulant
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Metaproterenol Sympathomimetic 2 adrenergic agonist Bronchodilator Used in asthma
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Metformin Oral hypoglycemic Biguanide Hepatic gluconeogenesis inhibitor
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Methacholine Cholinomimetic Bronchoconstrictor
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Methadone Opioid receptor agonist
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