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2004-2005 Pharmacology Review of Everything (Principles, Cardiovascular and Respiratory drugs have been updated) 19 December 2015 8:59 PM
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Methenamine Urinary tract antiseptic Decomposes to formaldehyde in acidic environment
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Methicillin Penicillin antibiotic Cell wall synthesis inhibitor Pencillinase resistant penicillin Inhibits peptidoglycan cross-linking
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Methimazol Antithyroid Prevents synthesis of thyroid hormones (blocks iodine organification)
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Methotrexate Immunosuppressive Antineoplastic Folic acid antagonist Dihydrofolate reductase inhibitor
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Methoxamine Sympathomimetic 1 adrenergic agonist Vasoconstrictor
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Methylcellulose Bulk laxative
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Methydopa Sympatholytic 2 adrenergic agonist Antihypertensive
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Methylphenidate Indirect sympathomimetic Drug of abuse ADD treatment Stimulant
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Methylprednisolone Adrenocorticosteroid Glucocorticoid Anti-inflammatory steroid Not by inhalation
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Methyltestosterone Androgen Synthetic oral
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Metipranolol Sympatholytic adrenergic antagonist Bronchoconstrictor
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Metoclopramide Prokinetic agent Antiemetic D 2 antagonist
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Metocurine Paralytic Paralyzes skeletal muscles
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Metolazone Thiazide-like diuretic Na-Cl symporter inhibitor Antihypertensive
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Metoprolol Sympatholytic 1 adrenergic antagonist Antihypertensive Heart failure medication Bronchoconstrictor
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Metronidazole Antibiotic Antiparasitic Antiulcer Anaerobes Reduction leads to intermediates that damage DNA
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Metyrapone Glucocorticoid antagonist
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Mexilitine Class I antiarrhythmic Na + channel blocker (activated and inactivated channels)
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Miconazole Imidazole antifungal Inhibits synthesis of ergosterol by inhibiting lanosterol 14 demethylase
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Midazolam Sedative hypnotic Short-acting benzodiazopine
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Mifepristone (RU-486) Progesterone antagonist
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Miglitol Oral hypoglycemic Alpha-glucosidase inhibitor Inhibits intestinal glucose absorption
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Mineral oil Lubricating laxative Stool softener
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Minocycline Tetracycline antibiotic Bacteriostatic protein synthesis inhibitor 30S ribosome Prevents aminoacyl tRNA attachment
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Minoxidil Vasodilator Antihypertensive
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Misoprostol Prostaglandin Antiulcer
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Mitomycin C Antineoplastic Natural product Antibiotic
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Mivacurium Paralytic Paralyzes skeletal muscles
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Moezipril Antihypertensive Converting enzyme inhibitor
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Montelukast Leukotriene inhibitor LTR1 and LTD4 antagonist Asthma treatment
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Moricizine Class I antiarrhythmic Na + channel blocker
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Morphine Opioid Analgesic receptor agonist
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Muromonab-CD3 Immunosuppressive Mouse monoclonal anti-CD3 antibody Organ transplant (anti-rejection)
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Mycophenolate Immunosuppressive Inhibits inosine monophosphate dehydrogenase activity
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Nadolol Sympatholytic adrenergic antagonist Antihypertensive
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Nafarelin Gonadotropin releasing hormone (GnRH) agonist
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Nafcillin Penicillin antibiotic Cell wall synthesis inhibitor Penicillinase resistant penicillin Inhibits peptidoglycan cross-linking
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Nalbuphine Opioid antagonist receptor antagonist
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Nalidixic acid Urinary tract antiseptic Quinolone Inhibits bacterial DNA gyrase
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Nalmefene Opioid antagonist
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Nalorphine Opioid antagonist
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Naloxone Opioid antagonist
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Naproxen NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Nateglinide Oral hypoglycemic Meglitinide Insulinotropic
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Naltrexone Opioid antagonist
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Nedocromil Mast cell stabilizer Inhibits release of mast cell mediators Used prophylactically in asthma
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Neomycin Aminoglycoside antibiotic Bactericidal protein synthesis inhibitor 30S ribosome Freezes initiation Topical
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Neostigmine Anticholinesterase Vasodilator Treatment for myaesthenia gravis Promotes defecation and urination Bronchoconstrictor
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Netilmicin Aminoglycoside antibiotic Bactericidal protein synthesis inhibitor 30S ribosome Freezes initiation
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Nevirapine Antiretroviral Non-nucleoside reverse transcriptase inhibitor (NNRTI)
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Nicardipine Antihypertensive Calcium channel blocker
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Nicotine Cholinomimetic Drug of abuse Nicotinic receptor agonist (skeletal muscle contraction) Stimulant Smoking cessation medication
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Nicotinic acid Antihyperlipidemic Inhibition of VLDL secretion (?)
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Nifedipine Antihypertensive Antianginal Calcium channel blocker
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Nifurtimox Tropical antiparasitic Treatment of South American Trypanosomiasis; Chagas disease
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Nisoldipine Antihypertensive Calcium channel blocker
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Nitrendipine Antihypertensive Calcium channel blocker
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Nitrofurantoin Urinary tract antiseptic Reduction leads to intermediates that damage DNA
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Nitroglycerine Venodilator Antianginal
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Nitroprusside Vasodilator Antihypertensive
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Nitrous oxide General anaesthetic Inhaled anaesthetic
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Nizatidine Antihistamine Antiulcer H 2 receptor antagonist
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Norepinephrine Sympathomimetic Vasoconstrictor
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Norethindrone Progestin 19-nor testosterone analogue Combination oral contraceptive
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Norethynodrel Progestin 19-nor testosterone analogue Combination oral contraceptive
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Norfloxacin Fluoroquinolone antibiotic DNA replication inhibitor Inhibits bacterial DNA gyrase
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Norgestimate Progestin 19-nor testosterone analogue Combination oral contraceptive
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Norgestrel Progestin 19-nor testosterone analogue Combination oral contraceptive
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Nortriptyline Tricyclic antidepressant (TCA)
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NPH insulin Hormone Insulin analogue Intermediate acting
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Non-steroidal Anti-inflammatory Drugs (NSAIDs) Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitors
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Nystatin Antifungal Polyene antibiotic Binds to ergosterol & alters permeability Topical
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Octreotide Somatostatin analogue Peptide hormone inhibitor Decreases growth hormone secretion Decreases gastric and pancreatic secretions
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Olsalazine NSAID (salicylate) Treatment of IBD
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Omeprazole/esomeprazole Antiulcer H + /K + ATPase inhibitor
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Ondansetron Antiemetic 5HT 3 receptor antagonist
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Organic antimonials Tropical antiparasitic Treatment of Leishmaniasis sodium stibogluconate meglumine antimonate
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Oseltamivir Antiviral Inhibits neuraminidase and decreases viral release Treatment of Influenza A & B
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Oxacillin Penicillin antibiotic Cell wall synthesis inhibitor Pencillinase resistant penicillin Inhibits peptidoglycan cross-linking
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Oxazepam Sedative/hypnotic Anxiolytic Benzodiazepine Acts on GABA A receptor complex
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Oxybutinin Anticholinergic Muscarinic receptor antagonist Prevents urination
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Oxycodone Analgesic Opioid agonist
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Oxytetracycline Tetracycline antibiotic Bacteriostatic protein synthesis inhibitor 30S ribosome Prevents aminoacyl tRNA attachment
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Oxytocin Hypothalamic (posterior pituitary) hormone Uterine stimulant
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Paclitaxel Antineoplastic Natural product Plant alkaloid (taxane)
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Palivizumab Antiviral Monoclonal antibody against the surface of respiratory syncytial virus
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Pamidronate Anti-osteoporesis Bisphosphonate Inhibitor of osteoclast-mediated bone resorption
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Pancuronium Paralytic Paralyzes skeletal muscles
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Pantoprazole Antiulcer H + /K + ATPase inhibitor
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Para-aminosalicylic acid Antibiotic Nucleic acid and protein synthesis inhibitor Inhibits dihydropteroate synthetase Secondary TB drug
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Paraldehyde Sedative/Hypnotic
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Parathyroid hormone Hormone Maintains plasma Ca 2+ concentrations
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Paromomycin Antiparasitic Aminoglycoside antibiotic Treatment of protozoal infections
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Pectin Antidiarrheal
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Penbutolol Sympatholytic adrenergic antagonist Antihypertensive Bronchoconstrictor
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Penciclovir Antiherpes Purine analog Phosphorylated to inhibitor of viral DNA polymerase
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Penicillins lactam antibiotics Cell wall synthesis inhibitors Inhibit cross-linking of peptidoglycan
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Penicillin G Penicillin antibiotic Cell wall synthesis inhibitor Acid labile Inhibits peptidoglycan cross-linking
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Penicillin V Penicillin antibiotic Cell wall synthesis inhibitor More acid resistant than Penicillin G Inhibits peptidoglycan cross-linking
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Pentamidine Tropical antiparasitic Treatment of African Trypanosomiasis
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