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2004-2005 Pharmacology Review of Everything (Principles, Cardiovascular and Respiratory drugs have been updated) 19 February 2016 2:39 PM
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Spectinomycin Antibiotic Bacteriostatic protein synthesis inhibitor 30S ribosome
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Spironolactone Potassium sparing diuretic Antiandrogen Aldosterone receptor antagonist Androgen receptor antagonist Testosterone synthesis inhibitor Antihypertensive Heart failure treatment
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St. John’s Wort Dietary supplement Antidepressant
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Streptokinase Thrombolytic
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Streptomycin Aminoglycoside antibiotic Bactericidal protein synthesis inhibitor 30S ribosome Freezes initiation
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Succinylcholine Paralytic Depolarizing blocker Paralyzes skeletal muscles Bronchoconstrictor
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Sucralfate Antiulcer
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Sufentanil Opioid General anaesthetic Intravenous anaesthetic
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Sulfacetamide Sulfonamide antibiotic Microbial nucleic acid and protein synthesis inhibitor Inhibits dihydropteroate synthetase Topical
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Sulfadoxine Sulfonamide antibiotic Microbial nucleic acid and protein synthesis inhibitor Dihydropteroate synthetase inhibitor
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Sulfamethoxazole Sulfonamide antibiotic Microbial nucleic acid and protein synthesis inhibitor Inhibits dihydropteroate synthetase
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Sulfasalazine Disease modifying anti-rheumatic drug (DMARD) Metabolized to sulfonamide + salicylate (NSAID) Treatment of IBD
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Sulfinpyrazone Uricosuric Anti-gout
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Sulfisoxazole Sulfonamide antibiotic Nucleic acid and protein synthesis inhibitor Inhibits dihydropteroate synthetase
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Sulfonamides Antibiotics Nucleic acid and protein synthesis inhibitors Inhibit dihydropteroate synthetase
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Sulindac NSAID Analgesic, Anti-inflammatory, Antipyretic Cyclooxygenase inhibitor
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Suramin Tropical antiparasitic Treatment of African Trypanosomiasis
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Tacrolimus Immunosuppressive Antineoplastic Binds FKBP (FK506 binding protein) Inhibits calcineurin
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Tamoxifen Antineoplastic Antiestrogen Estrogen receptor anatagonist
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Tegaserod IBS treatment 5HT 4 receptor agonist
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Telmisartan Antihypertensive Angiotensin receptor blocker (ARB)
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Temazepam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
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Tenecteplase Thrombolytic Tissue plasminogen activator (tPA)
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Terazosin Sympatholytic 1 adrenergic antagonist Antihypertensive Treatment for benign prostatic hypertrophy
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Terbinafine Allylamine antifungal Inhibits ergosterol synthesis by inhibiting squalene epoxidase
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Terbutaline Sympathomimetic 2 adrenergic agonist Short acting bronchodilator Tocolytic Uterine relaxant
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Testosterone Androgen Natural male gonadal steroid
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Testosterone cypionate Androgen Synthetic depot
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Testosterone enanthate Androgen Synthetic depot
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Testosterone propionate Androgen Synthetic depot
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Tetracaine Local anaesthetic
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Tetracycline Antibiotic Bacteriostatic protein synthesis inhibitor Antiulcer 30S ribosome Prevents aminoacyl tRNA attachment
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Thalidomide Antineoplastic Leprosy treatment Anti-angiogenic Anti-TNF
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Theophylline Bronchodilator Methylxanthine Phosphodiesterase inhibitor Used in asthma
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Thiabendazole Antihelminthic Treatment of intestinal roundworms
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6-Thioguanine Antineoplastic Antimetabolite (“pseudofeedback inhibition” of HGPRT and PRP – purine synthesis)
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Thiopental General Anaesthetic Ultra-short-acting barbiturate
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Thioridazine Antipsychotic Phenothiazine
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Thiotepa Antineoplastic Alkylating agent
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Thiothixene Antipsychotic
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Thrombopoietin Cytokine Platelet synthesis stimulator
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Thromboxane A 2 (TXA 2 ) Autacoid Promotes platelet aggregation Cyclooxygenase product of arachidonate metabolism
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Thyrotropin-releasing Hormone (TRH) Hypothalamic hormone Stimulates release of thyroid stimulating hormone (TSH) from the anterior pituitary
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Thyrotropin Thyroid-stimulating Hormone (TSH) Anterior pituitary hormone Stimulates production of thyroxine (T 4 ), triiodothyronine (T 3 ) and thyroglobulin
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Ticarcillin Penicillin antibiotic Cell wall synthesis inhibitor Anti-pseudomonal penicillin Inhibits peptidoglycan cross-linking
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Ticlopidine Antiplatelet ADP receptor antagonist
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Timolol Sympatholytic adrenergic antagonist Antihypertensive Glaucoma treatment Anti-anginal Bronchoconstrictor
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Tissue plasminogen activators Thrombolytics alteplase, reteplase, tenecteplase
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Tobramycin Aminoglycoside antibiotic Bactericidal protein synthesis inhibitor 30S ribosome Freezes initiation
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Tocainide Class I antiarrhythmic Na + channel blocker (activated channels)
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Tolbutamide Oral hypoglycemic Sulfonylurea Insulinotropic
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Tolterodine Anticholinergic Muscarinic receptor antagonist Prevents urination
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Toremifene Estrogen antagonist Selective estrogen receptor modulator (SERM)
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Tosemide Loop diuretic Na-K-2Cl symporter inhibitor
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Trandopril Antihypertensive Converting enzyme inhibitor
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Tranylcypromine Antidepressant Monoamine oxidase inhibitor (MAO-I)
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Trastuzumab Antineoplastic Anti-HER2 antibody
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Triamcinolone Adrenocorticosteroid Glucocorticoid Anti-inflammatory steroid Inhaled
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Triamterene Potassium sparing diuretic Sodium channel inhibitor Antihypertensive
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Triazolam Sedative/Hypnotic Benzodiazepine Acts on GABA A receptor complex
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Trifluoperazine Antipsychotic Phenothiazine
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Trifluridine Antiherpes Pyrimidine analog Phosphorylated to inhibitor of viral DNA polymerase
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Trihexyphenidyl Antiparkinson Antimuscarinic
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Trimethaphan Sympatholytic Anticholinergic Nicotinic antagonist Antihypertensive
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Trimethoprim Antibiotic Protein and nucleic acid synthesis inhibitor Inhibits bacterial dihydrofolate reductase
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Tripelennamine Classical antihistamine H 1 antagonist
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Tubocurarine Paralytic Paralyzes skeletal muscles
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Tumor necrosis factor Cytokine Antineoplastic
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Tyramine Indirect sympathomimetic Vasoconstrictor Vasopressor
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Ultralente insulin Hormone Insulin analogue Long acting
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Urokinase Thrombolytic
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Valacyclovir Antiherpes Purine analog Phosphorylated to inhibitor of viral DNA polymerase
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Valsartan Antihypertensive Angiotensin receptor blocker (ARB)
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Valganciclovir Antiherpes Purine analog Phosphorylated to inhibitor of viral DNA polymerase
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Valproic acid Anticonvulsant
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Valsartan Antihypertensive Angiotensin receptor blocker (ARB)
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Vancomycin Antibiotic Inhibits cell wall synthesis Not a lactam
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Arginine vasopressin (Antidiuretic hormone; ADH) Hypothalamic (posterior pituitary) hormone Antidiuretic Vasoconstrictor
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Vecuronium Paralytic Paralyze skeletal muscles
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Verapamil Class IV antiarrhythmic Antihypertensive L-type Ca 2+ channel blocker Antianginal
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Vigabatrin Anticonvulsant Irreversible GABA aminotransferase inhibitor
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Vinblastine Antineoplastic Vinca alkaloid Natural product
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Vincristine Antineoplastic Vinca alkaloid Natural product
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Voriconazole Triazole antifungal Inhibits synthesis of ergosterol by inhibiting lanosterol 14 demethylase
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Warfarin Anticoagulant Vitamin K synthesis inhibitor
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Zafirlukast Leukotriene inhibitor LTR 1 and LTD 4 antagonist Asthma treatment
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Zalcitabine Antiretroviral Nucleoside reverse transcriptase inhibitor (NRTI) Dideoxycytidine (ddC)
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Zanamivir Antiviral Inhibits neuraminidase and decreases viral release Treatment of Influenza A & B
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Zidovudine Antiretroviral Nucleoside reverse transcriptase inhibitor (NRTI) Azidothymidine (AZT)
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Zileuton Leukotriene inhibitor 5-lipoxygenase inhibitor Used in asthma
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Zolpidem Sedative/Hypnotic Non-benzodiazepine
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